Aminoglycoside antibiotics are important for treating serious bacterial infections. A number of advances in their chemistry, biochemistry and recognition have come about in the last ten-fifteen years which have led to the development of novel antibiotics and opened up new therapeutic targets for intervention. Addressing the chemistry, biology, and toxicology of aminoglycosides, Aminoglycoside Antibiotics: From Chemical Biology to Drug Discovery brings professionals and students in the field up to date on these advances in the field and helps them fulfill the enormous potential of aminoglycodises for drug discovery and rational drug design.